Publications 2017


  • Bioinorganic Chemistry

Sensitivity towards the GRP78 inhibitor KP1339/IT-139 is characterized by apoptosis induction via caspase 8 upon disruption of ER homeostasis
Schoenhacker-Alte, B., Mohr, T., Pirker, C., Kryeziu, K., Kuhn, P-S., Buck, A., Hofmann, T., Gerner, C., Hermann, G., Koellensperger, G., Keppler, B. K., Berger, W. & Heffeter, P.
Cancer Letters (2017) 404, 79-88

Synthesis and in vivo anticancer evaluation of poly(organo) phosphazene-based metallodrug conjugates
Hackl, C. M., Schoenhacker-Alte, B., Klose, M. H. M., Henke, H., Legina, M. S., Jakupec, M. A., Berger, W., Keppler, B. K., Brueggemann, O., Teasdale, I., Heffeter, P. & Kandioller, W.
Dalton Transactions (Print Edition): a journal of inorganic chemistry (2017) 46, 36, 12114-12124

Fast High-Resolution Laser Ablation-Inductively Coupled Plasma Mass Spectrometry Imaging of the Distribution of Platinum-Based Anticancer Compounds in Multicellular Tumor Spheroids
Theiner, S., Van Malderen, S. J. M., Van Acker, T., Legin, A., Keppler, B. K., Vanhaecke, F. & Koellensperger
Analytical Chemistry (2017) 89, 23, 12641-12645

A fluorescent oxaliplatin derivative for investigation of oxaliplatin resistance using imaging techniques
Kalayda, G. V., Kullmann, M., Galanski, M. & Gollos
Journal of Biological Inorganic Chemistry (2017) 22, 8, 1295-1304

Optically active histidin-2-ylidene stabilised gold nanoparticles
Young, A. J., Serpell, C. J., Chin, J. M. & Reithofer, M. R.
Chemical Communications  (2017) 53, 92, 12426-12429

Magnetic Control of MOF Crystal Orientation and Alignment
Cheng, F., Marshall, E. S., Young, A. J., Robinson, P. J., Bouillard, J-S. G., Adawi, A. M., Vermeulen, N. A., Farha, O. K., Reithofer, M. R. & Chin, J. M.
Chemistry: A European Journal (2017) 23, 62, 15578-15582

Effects of Terminal Substitution and Iron Coordination on Antiproliferative Activity of l-Proline-salicylaldehyde-Thiosemicarbazone Hybrids
Milunovic, M. N. M., Dobrova, A., Novitchi, G., Gligorijevic, N., Radulovic, S., Kozisek, J., Rapta, P., Enyedy, E. A. & Arion, V. B.
European Journal of Inorganic Chemistry  (2017) 40, 4773-4783

A Bis(mu-chlorido)-Bridged Cobalt(II) Complex with Silyl-Containing Schiff Base as a Catalyst Precursor in the Solvent-Free Oxidation of Cyclohexane
Zaltariov, M-F., Vieru, V., Zalibera, M., Cazacu, M., Martins, N. M. R., Martins, L. M. D. R. S., Rapta, P., Novitchi, G., Shova, S., Pombeiro, A. J. L. & Arion, V. B.
European Journal of Inorganic Chemistry (2017) 37, 4324-4332

Comparative equilibrium and structural studies of new pentamethylcyclopentadienyl rhodium complexes bearing (O, N) donor bidentate ligands
Domotor, O., Hackl, C. M., Bali, K., Roller, A., Hejl, M., Jakupec, M. A., Keppler, B. K., Kandioller, W. & Enyedy, E. A.
Journal of Organometallic Chemistry (2017) 846, 287-295

A five-coordinate manganese(III) complex of a salen type ligand with a positive axial anisotropy parameter D
Shova, S., Vlad, A., Cazacu, M., Krzystek, J., Bucinsky, L., Breza, M., Darvasiova, D., Rapta, P., Cano, J., Telser, J. & Arion, V. B.
Dalton Transactions (Print Edition) (2017) 46, 35, 11817-11829

cis-Tetrachlorido-bis(indazole)osmium(IV) and its osmium(III) analogues: paving the way towards the cis-isomer of the ruthenium anticancer drugs KP1019 and/or NKP1339
Buchel, G. E., Kossatz, S., Sadique, A., Rapta, P., Zalibera, M., Bucinsky, L., Komorovsky, S., Telser, J., Eppinger, J., Reiner, T. & Arion, V. B.
Dalton Transactions (Print Edition) (2017) 46, 35, 11925-11941

Platinum(IV) Complexes Featuring Axial Michael Acceptor Ligands - Synthesis, Characterization, and Cytotoxicity
Sommerfeld, N. S., Strohhofer, D., Cseh, K., Theiner, S., Jakupec, M. A., Koellensperger, G., Galanski, M. & Keppler, B. K.
European Journal of Inorganic Chemistry (2017) 34, 4049-4054

Intrinsic fluorescence of the clinically approved multikinase inhibitor nintedanib reveals lysosomal sequestration as resistance mechanism in FGFR-driven lung cancer
Englinger, B., Kallus, S., Senkiv, J., Heilos, D., Gabler, L., Van Schoonhoven, S., Terenzi, A., Moser, P., Pirker, C., Timelthaler, G., Jaeger, W., Kowol, C. R., Heffeter, P., Grusch, M. & Berger, W.
Journal of Experimental and Clinical Cancer Research  (2017) 36, 122

Understanding the metabolism of the anticancer drug Triapine: electrochemical oxidation, microsomal incubation and in vivo analysis using LC-HRMS
Pelivan, K., Frensemeier, L., Karst, U., Koellensperger, G., Bielec, B., Hager, S., Heffeter, P., Keppler, B. K. & Kowol, C. R.
The Analyst (2017) 142, 17, 3165-3176

Impact of the equatorial coordination sphere on the rate of reduction, lipophilicity and cytotoxic activity of platinum(IV) complexes
Hoefer, D., Varbanov, H. P., Hejl, M., Jakupec, M. A., Roller, A., Galanski, M. & Keppler, B. K.
Journal of Inorganic Biochemistry (2017) 174, 119-129

Multifunctional alpha(v)beta(6) Integrin-Specific Peptide-Pt(IV) Conjugates for Cancer Cell Targeting
Conibear, A. C., Hager, S., Mayr, J., Klose, M. H. M., Keppler, B. K., Kowol, C. R., Heffeter, P. & Becker, C. F. W.
Bioconjugate Chemistry (2017) 28, 9, 2429-2439

Self-Ordering Secondary Structure of D- and L-Arginine-Derived Polyamidoamino Acids
Manfredi, A., Mauro, N., Terenzi, A., Alongi, J., Lazzari, F., Ganazzoli, F., Raffaini, G., Ranucci, E. & Ferruti, P.
ACS Macro Letters (2017) 6, 9, 987-991

Electronic State of Sodium trans-[Tetrachloridobis(1H-indazole)ruthenate(III)] (NKP-1339) in Tumor, Liver and Kidney Tissue of a SW480-bearing Mouse
Blazevic, A., Hummer, A. A., Heffeter, P., Berger, W., Filipits, M., Cibin, G., Keppler, B. K. & Rompel, A.
Scientific Reports
(2017) 7, 40966

Introducing the 4-Phenyl-1,2,3-Triazole Moiety as a Versatile Scaffold for the Development of Cytotoxic Ruthenium(II) and Osmium(II) Arene Cyclometalates
Riedl, C. A., Flocke, L. S., Hejl, M., Roller, A., Klose, M. H. M., Jakupec, M. A., Kandioller, W. & Keppler, B. K.
Inorganic Chemistry
(2017) 56, 1, 528-541

An iron(III)-centred ferric wheel Fe subset of{Fe-6} with a siloxane-based bis-salicylidene Schiff base
Shova, S., Cazacu, M., Novitchi, G., Zoppellaro, G., Train, C. & Arion, V. B.
Dalton Transactions
(2017) 46, 6, 1789-1793

Comparative studies of oxaliplatin-based platinum(IV) complexes in different in vitro and in vivo tumor models
Goeschl, S., Schreiber-Brynzak, E., Pichler, V., Cseh, K., Heffeter, P., Jungwirth, U., Jakupec, M. A., Berger, W. & Keppler, B. K.
(2017) 9, 3, 309-322

Copper(ii) thiosemicarbazone complexes induce marked ROS accumulation and promote nrf2-mediated antioxidant response in highly resistant breast cancer cells
Sîrbu, A., Palamarciuc, O., Babak, M. V., Lim, J. M., Ohui, K., Enyedy, E. A., Shova, S., Darvasiová, D., Rapta, P., Ang, W. H. & Arion, V. B.
Dalton Transactions
(2017) 46, 12, 3833-3847

Influence of the Number of Axial Bexarotene Ligands on the Cytotoxicity of Pt(IV) Analogs of Oxaliplatin
Nosova, Y. N., Zenin, I. V., Maximova, V. P., Zhidkova, E. M., Kirsanov, K. I., Lesovaya, E. A., Lobas, A. A., Gorshkov, M. V., Kovaleva, O. N., Milaeva, E. R., Galanski, M., Keppler, B. K. & Nazarov, A. A.
Bioinorganic Chemistry and Applications
(2017) 4736321

Response Profiling Using Shotgun Proteomics Enables Global Metallodrug Mechanisms of Action To Be Established
Kreutz, D., Bileck, A., Plessl, K., Wolrab, D., Groessl, M., Keppler, B. K., Meier, S. M. & Gerner, C.
Chemistry: A European Journal
(2017) 23, 8, S. 1881-1890

Self-assembled Pt2L2 boxes strongly bind G-quadruplex DNA and influence gene expression in cancer cells
Domarco, O., Loetsch, D., Schreiber, J., Dinhof, C., Van Schoonhoven, S., Garcia, M. D., Peinador, C., Keppler, B. K., Berger, W. & Terenzi, A.
Dalton Transactions (Print Edition)
(2017) 46, 2, 329-332

Characterizing activation mechanisms and binding preferences of ruthenium metallo-prodrugs by a competitive binding assay
Artner, C., Holtkamp, H. U., Hartinger, C. G. & Meier-Menches, S. M.

Journal of Inorganic Biochemistry (2017) 177, 322-327

Metal NHC Complexes with Naphthalimide Ligands as DNA-Interacting Antiproliferative Agents
Streciwilk, W., Terenzi, A., Misgeld, R., Frias, C., Jones, P. G., Prokop, A., Keppler, B. K. & Ott, I.
(2017) 12, 3, 214-225

Complex formation reactions of gallium(III) and iron(III/II) with L-proline-thiosemicarbazone hybrids: A comparative study
Bacher, F., Domotor, O., Enyedy, E. A., Filipovic, L., Radulovic, S., Smith, G. S. & Arion, V.
Inorganica Chimica Acta
(2017) 455, 505-513

Oxaliplatin reacts with DMSO only in the presence of water
Varbanov, H. P., Ortiz, D., Hoefer, D., Menin, L., Galanski, M., Keppler, B. K. & Dyson, P. J.
Dalton Transactions (Print Edition)
(2017) 46, 28, 8929-8932

Amidoxime platinum(II) complexes: pH-dependent highly selective generation and cytotoxic activity
Bolotin, D. S., Demakova, M. Y., Legin, A. A., Suslonov, V. V., Nazarov, A. A., Jakupec, M. A., Keppler, B. K. & Kukushkin, V. Y.
New Journal of Chemistry
(2017) 41, 14, 6840-6848

Conversion of hydrazides into N,N '-diacylhydrazines in the presence of a ruthenium(II)-arene complex
Nikolic, S., Ciric, I., Roller, A., Lukes, V., Arion, V. B. & Grguric-Sipka, S.
New Journal of Chemistry
(2017) 41, 14, 6857-6865

DNA or protein? Capillary zone electrophoresismass spectrometry rapidly elucidates metallodrug binding selectivity
Artner, C., Holtkamp, H. U., Kandioller, W., Hartinger, C. G., Meier, S. M. & Keppler, B. K.
Chemical Communications
(2017) 53, 57, 8002-8005

Post-digestion stabilization of osmium enables quantification by ICP-MS in cell culture and tissue
Klose, M. H. M., Hejl, M., Heffeter, P., Jakupec, M. A., Meier, S. M., Berger, W. & Keppler, B. K.
The Analyst
(2017) 142, 13, 2327-2332

An Organoruthenium Anticancer Agent Shows Unexpected Target Selectivity For Plectin
Meier, S. M., Kreutz, D., Winter, L., Klose, M. H. M., Cseh, K., Weiss, T., Bileck, A., Alte, B., Mader, J. C., Jana, S., Chatterjee, A., Bhattacharyya, A., Hejl, M., Jakupec, M. A., Heffeter, P., Berger, W., Hartinger, C. G., Keppler, B. K., Wiche, G. & Gerner, C.
Angewandte Chemie (International Edition) (2017) 56, 28, 8267-8271

Antiproliferative Copper(II) and Platinum(II) Complexes with Bidentate N,N-Donor Ligands
Sommerfeld, N. S., Guelzow, J., Roller, A., Cseh, K., Jakupec, M. A., Grohmann, A., Galanski, M. & Keppler, B. K.
European Journal of Inorganic Chemistry
(2017) 24, 3115-3124

On the nature of photoluminescence in Bismuth-doped silica glass
Laguta, O. V., El Hamzaoui, H., Bouazaoui, M., Arion, V. B. & Razdobreev, I. M.
Scientific Reports
(2017) 7, 3178

EGFR-targeting peptide-coupled platinum(IV) complexes
Mayr, J., Hager, S., Koblmueller, B., Klose, M. H. M., Holste, K., Fischer, B., Pelivan, K., Berger, W., Heffeter, P., Kowol, C. R. & Keppler, B. K.
Journal of Biological Inorganic Chemistry
(2017) 22, 4, 591-603

Functionalization of Ruthenium(II)(eta(6)-p-cymene)(3-hydroxy-2-pyridone) Complexes with (Thio)Morpholine: Synthesis and Bioanalytical Studies
Hanif, M., Meier, S. M., Adhireksan, Z., Henke, H., Martic, S., Movassaghi, S., Labib, M., Kandioller, W., Jamieson, S. M. F., Hejl, M., Jakupec, M. A., Kraatz, H-B., Davey, C. A., Keppler, B. K. & Hartinger, C. G.
(2017) 82, 6, 841-847

Synthesis, Characterization, and Time-Dependent NMR Spectroscopy Studies of (SP-4-2)-[(trans-1R,2R/1S,2S-N-15(2))-Cyclohexane-1,2-diamine][(C-13(2))oxalato]platinum(II)
Hoefer, D., Galanski, M. & Keppler, B. K.

European Journal of Inorganic Chemistry
(2017) 17, 2347-2354

Rapid generation of hydrogen peroxide contributes to the complex cell death induction by the angucycline antibiotic landomycin E
Panchuk, R. R., Lehka, L. V., Terenzi, A., Matselyukh, B. P., Rohr, J., Jha, A. K., Downey, T., Kril, I. J., Herbacek, I., Schoonhoven, S., Heffeter, P., Stoika, R. S. & Berger, W.
Free Radical Biology & Medicine
(2017) 106, 134-147

Distinct activity of the bone-targeted gallium compound KP46 against osteosarcoma cells - synergism with autophagy inhibition
Kubista, B., Schoefl, T., Mayr, L., van Schoonhoven, S., Heffeter, P., Windhager, R., Keppler, B. K. & Berger, W.
Journal of Experimental and Clinical Cancer Research
(2017) 36, 52

{Ru(CO)(x)}-Core complexes with benzimidazole ligands: synthesis, X-ray structure and evaluation of anticancer activity in vivo
Tamasi, G., Merlino, A., Scaletti, F., Heffeter, P., Legin, A. A., Jakupec, M. A., Berger, W., Messori, L., Keppler, B. K. & Cini, R.
Dalton Transactions (Print Edition)
(2017) 46, 9, 3025-3040

An albumin-based tumor-targeted oxaliplatin prodrug with distinctly improved anticancer activity in vivo
Mayr, J., Heffeter, P., Groza, D., Galvez, L., Koellensperger, G., Roller, A., Alte, B., Haider, M., Berger, W., Kowol, C. R. & Keppler, B. K.
Chemical Science
(2017) 8, 3, 2241-2250

Loss of CUL4A expression is underlying cisplatin hypersensitivity in colorectal carcinoma cells with acquired trabectedin resistance
Englinger, B., Mair, M., Miklos, W., Pirker, C., Mohr, T., van Schoonhoven, S., Loetsch, D., Körner, W., Ferk, F., Knasmueller, S., Heffeter, P., Keppler, B. K., Grusch, M. & Berger, W.
British Journal of Cancer
(2017) 116, 4, 489-500

Application of imaging mass spectrometry approaches to facilitate metal-based anticancer drug research
Lee, R. F. S., Theiner, S., Meibom, A., Koellensperger, G., Keppler, B. K. & Dyson, P. J.
(2017) 9, 4, 365-381

Enhancing the Cytotoxic Activity of Anticancer Pt-IV Complexes by Introduction of Lonidamine as an Axial Ligand
Nosova, Y. N., Foteeva, L. S., Zenin, I. V., Fetisov, T. I., Kirsanov, K. I., Yakubovskaya, M. G., Antonenko, T. A., Tafeenko, V. A., Aslanov, L. A., Lobas, A. A., Gorshkov, M. V., Galanski, M., Keppler, B. K., Timerbaev, A. R., Milaeva, E. R. & Nazarov, A. A.
European Journal of Inorganic Chemistry
(2017) 12, 1785-1791

Low-Generation Polyamidoamine Dendrimers as Drug Carriers for Platinum(IV) Complexes
Sommerfeld, N. S., Hejl, M., Klose, M. H. M., Schreiber-Brynzak, E., Bileck, A., Meier, S. M., Gerner, C., Jakupec, M. A., Galanski, M. & Keppler, B. K.
European Journal of Inorganic Chemistry
(2017) 12, 1713-1720

New Iminodiacetate -Thiosemicarbazone Hybrids and Their Copper(II) Complexes Are Potential Ribonucleotide Reductase R2 Inhibitors with High Antiproliferative Activity
Zaltariov, M. F., Hammerstad, M., Arabshahi, H. J., Jovanovic, K., Richter, K. W., Cazacu, M., Shova, S., Balan, M., Andersen, N. H., Raduloyic, S., Reynisson, J., Andersson, K. & Arion, V. B.
Inorganic Chemistry (2017) 56, 6, 3532-3549

  • Environmental Chemistry and Radiochemistry

beta-O-4 type dilignol compounds and their iron complexes for modeling of iron binding to humic acids: synthesis, characterization, electrochemical studies and algal growth experiments
Orlowska, E., Enyedy, E. A., Pignitter, M., Jirsa, F., Krachler, R., Kandioller, W. & Keppler, B. K.
New Journal of Chemistry (2017) 41, 20, 11546-11555

Thioglycolate-based task-specific ionic liquids: Metal extraction abilities vs acute algal toxicity
Platzer, S., Leyma, R., Wolske, S., Kandioller, W., Heid, E., Schroeder, C., Schagerl, M., Krachler, R., Jirsa, F. & Keppler, B. K.
Journal of Hazardous Materials (2017) 340, 113-119

Fish as bioindicators for trace element pollution from two contrasting lakes in the Eastern Rift Valley, Kenya: spatial and temporal aspects
Plessl, C., Otachi, E. O., Koerner, W., Avenant-Oldewage, A. & Jirsa, F.
Environmental Science and Pollution Research
(2017) 24, 24, 19767-19776

Evaluation of Trace Element and Metal Accumulation and Edibility Risk Associated with Consumption of Labeo umbratus from the Vaal Dam, South Africa
Gilbert, B. M., Hussain , E., Jirsa, F. & Avenant-Oldewage,
International Journal of Environmental Research and Public Health
(2017) 14, 7, 678

Heavy metals in the mallard Anas platyrhynchos from eastern Austria
Plessl, C., Jandrisits, P., Krachler, R., Keppler, B. K. & Jirsa, F.
Science of the Total Environment
(2017) 580, 670-676

Task-specific thioglycolate ionic liquids for heavy metal extraction: Synthesis, extraction efficacies and recycling properties
Platzer, S., Kar, M., Leyma, R., Chib, S., Roller, A., Jirsa, F., Krachler, R., MacFarlane, D. R., Kandioller, W. & Keppler, B. K.
Journal of Hazardous Materials (2017) 324, Part B, 241-249

Synthetic iron complexes as models for natural iron-humic compounds: Synthesis, characterization and algal growth experiments
Orlowska, E., Roller, A., Pignitter, M., Jirsa, F., Krachler, R., Kandioller, W. & Keppler, B. K.
Science of the Total Environment
(2017) 577, 94-104

From the peat bog to the estuarine mixing zone: Common features and variances in riverine dissolved organic matter determined by non-targeted analysis
Rathgeb, A., Causon, T., Krachler, R. & Hann, S.
Marine Chemistry (2017) 194, 158-167

Development of a radiolabeled caninized anti-EGFR antibody for comparative oncology trials
Fazekas-Singer, J., Berroteran-Infante, N., Rami-Mark, C., Dumanic, M., Matz, M., Willmann, M., Andreae, F., Singer, J., Wadsak, W., Mitterhauser, M. & Jensen-Jarolim, E.
Onco Target  (2017) 8, 47, 83128-83141

In vivo evaluation of radiotracers targeting the melanin-concentrating hormone receptor 1: [C-11]SNAP-7941 and [F-18]FE@SNAP reveal specific uptake in the ventricular system
Zeilinger, M., Dumanic, M., Pichler, F., Budinsky, L., Wadsak, W., Pallitsch, K., Spreitzer, H., Hacker, M., Mitterhauser, M. & Philippe, C.
Scientific Reports (2017) 7, 10, 8054

LogP, a yesterday's value?
Vraka, C., Nics, L., Wagner, K-H., Hacker, M., Wadsak, W. & Mitterhauser, M.
Nuclear Medicine and Biology (2017) 50, 1-10

New approaches for the reliable in vitro assessment of binding affinity based on high-resolution real-time data acquisition of radioligand-receptor binding kinetics
Zeilinger, M., Pichler, F., Nics, L., Wadsak, W., Spreitzer, H., Hacker, M. & Mitterhauser, M.
EJNMMI Research (2017) 7, 22

  • Nucleic Acid Chemistry

High-Power 365 nm UV LED Mercury Arc Lamp Replacement for Photochemistry and Chemical Photolithography
Hölz, K., Lietard, J. & Somoza, M. M.
ACS Sustainable Chemistry & Engineering
(2017) 5, 1, 828-834

Mapping the affinity landscape of Thrombin-binding aptamers on 2 ' F-ANA/DNA chimeric G-Quadruplex microarrays
Lietard, J., Abou Assi, H., Gomez-Pinto, I., Gonzalez, C., Somoza, M. M. & Damha, M. J.
Nucleic Acids Research
(2017) 45, 4, 1619-1632

Hamming Distance as a Concept in DNA Molecular Recgonition
Mohammadi-Kambs, M., Hölz, K., Somoza, M. M. & Ott, A.
ACS Omega
(2017) 2, 4, 1302-1308

In vitro combinatory effects of the Alternaria mycotoxins alternariol and altertoxin II and potentially involved miRNAs
Vejdovszky, K., Sack, M., Jarolim, K., Aichinger, G., Somoza, M. M. & Marko, D.
Toxicology Letters
(2017) 267, 45-52

Caffeine induces gastric acid secretion via bitter taste signaling in gastric parietal cells
Liszt, K. I., Ley, J. P., Lieder, B., Behrens, M., Stoeger, V., Reiner-Concin, A., Hochkogler, C. M., Koeck, E., Marchiori, A., Hans, J., Widder, S., Krammer, G., Sanger, G. J., Somoza, M. M., Meyerhof, W. & Somoza, V.
Proceedings of the National Academy of Sciences of the United States of America (PNAS) 
(2017) 114, 30, E6260-E6269

  • X-ray Structure Analysis Centre

Heterocyclic Analogues of Modafinil as Novel, Atypical Dopamine Transporter Inhibitors
Kalaba, P., Aher, N. Y., Ilic, M., Dragacevic, V., Wieder, M., Miklosi, A. G., Zehl, M., Wackerlig, J., Roller, A., Beryozkina, T., Radoman, B., Saroja, S. R., Lindner, W., Gonzalez, E. P., Bakulev, V., Leban, J. J., Sitte, H. H., Urban, E., Langer, T. & Lubec, G.
Journal of Medicinal Chemistry (2017) 60, 22, 9330-9348

C2-Modified Sparteine Derivatives Are a New Class of Potentially Long-Acting Sodium Channel Blockers
Gawali, V. S., Simeonov, S., Drescher, M., Knott, T., Scheel, O., Kudolo, J., Kählig, H., Hochenegg, U., Roller, A., Todt, H. & Maulide, N.
ChemMedChem (2017) 12, 22, 1819–1822

Chemical Synthesis of (R-P)- and (S-P)-[O-16,O-17,O-18]Phosphoenol Pyruvate
Krizkova, P. M., Prechelmacher, S., Roller, A. & Hammerschmidt, F.
The Journal of Organic Chemistry (2017) 82, 19, 10310-10318

Synthesis of tetrasubstituted pyrazoles containing pyridinyl substituents
Jansa, J., Schmidt, R., Mamuye, A. D., Castoldi, L., Roller, A., Pace, V. & Holzer, W.
Beilstein Journal of Organic Chemistry 
(2017) 13, 895-902

Synthesis and antimicrobial evaluation of novel analogues of dehydroabietic acid prepared by C-H-Activation
Berger, M., Roller, A. & Maulide, N.
European Journal of Medicinal Chemistry
(2017) 126, 937-943

A greener and efficient access to substituted four- and six-membered sulfur-bearing heterocycles
Parisi, G., Degennaro, L., Carlucci, C., de Candia, M., Mastrorilli, P., Roller, A., Holzer, W., Altomare, C. D., Pace, V. & Luisi, R.

Organic & Biomolecular Chemistry
(2017) 12, 23, 5000-5015

A Methylidene Group in the Phosphonic Acid Analogue of Phenylalanine Reverses the Enantiopreference of Binding to Phenylalanine Ammonia-Lyases
Bata, Z., Qian, R., Roller, A., Horak, J., Bencze, L. C., Paizs, C., Hammerschmidt, F., Vertessy, B. G. & Poppe, L.
Advanced Synthesis & Catalysis
(2017) 359, 12, 2109-2120

Towards the biodegradation pathway of fosfomycin
Pallitsch, K., Schweifer, A., Roller, A. & Hammerschmidt, F.
Organic & Biomolecular Chemistry
(2017) 15, 15, 3276-3285