Fluorescence properties and cellular distribution of the investigational anticancer drug Triapine (3-aminopyridine-2-carboxaldehyde thiosemicarbazone) and its zinc(II) complex)

Author(s)
Christian Kowol, Robert Trondl, Vladimir Arion, Michael Jakupec, Irene Lichtscheidl-Schultz, Bernhard Keppler
Abstract

Triapine (3-aminopyridine-2-carboxaldehyde thiosemicarbazone), which entered several phase I and II clinical trials as an antitumor chemotherapeutic agent, was found to possess intrinsic fluorescence properties (lambda(ex) = 360 nm), which enabled us to monitor the uptake and intracellular distribution in living human cancer cells by fluorescence microscopy.

Organisation(s)
Department of Inorganic Chemistry
Journal
Dalton Transactions
Volume
39
Pages
704-706
No. of pages
3
ISSN
1477-9226
DOI
https://doi.org/10.1039/b919119b
Publication date
2010
Peer reviewed
Yes
Austrian Fields of Science 2012
1040 Chemistry
Sustainable Development Goals
SDG 3 - Good Health and Well-being
Portal url
https://ucrisportal.univie.ac.at/en/publications/74f9da5e-1557-4f13-b3a9-8c9a0b344d2e