Geminal homologative fluorination of carbonyl derivatives <i>en route</i> to 1-fluoro-2-haloethyl skeletons

Author(s)
Margherita Miele, Davide Castiglione, Alexander Prado-Roller, Laura Castoldi, Vittorio Pace
Abstract

Carbonyl groups undergo the sequential installation of two nucleophilic elements, halomethyl and fluoride moieties. This formal gem-difunctionalization enables the preparation-under full chemocontrol - of vic-fluorohaloethanes by simply defining the C1 nucleophile, thus enabling access to all combinations of the four halogens.

Organisation(s)
Core Facility Crystal Structure Analysis, Department of Inorganic Chemistry
External organisation(s)
University of Turin, Università degli Studi di Milano
Journal
Chemical Communications
ISSN
1359-7345
DOI
https://doi.org/10.1039/d5cc01542a
Publication date
06-2025
Peer reviewed
Yes
Austrian Fields of Science 2012
104015 Organic chemistry
ASJC Scopus subject areas
Electronic, Optical and Magnetic Materials, General Chemistry, Ceramics and Composites, Metals and Alloys, Materials Chemistry, Surfaces, Coatings and Films, Catalysis
Portal url
https://ucrisportal.univie.ac.at/en/publications/94563877-afe9-4fbb-8719-7216b2de295f