o. Univ.-Prof. Dr. Dr. Bernhard Keppler

Email: bernhard.keppler@univie.ac.at
Phone: +43-1-4277-52602

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Publications


Estrone-salicylaldehyde N-methylated thiosemicarbazone hybrids and their copper complexes: solution structure, stability and anticancer activity in tumour spheroids. / Petrasheuskaya, Tatsiana V.; Wernitznig, Debora; Kiss, Marton A. et al.
In: Journal of Biological Inorganic Chemistry, Vol. 26, No. 7, 10.2021, p. 775–791.

Publications: Contribution to journalArticlePeer Reviewed


Liposomal formulations of anticancer copper(ii) thiosemicarbazone complexes. / Mathuber, Marlene; Hager, Sonja; Keppler, Bernhard K. et al.
In: Dalton Transactions, Vol. 50, No. 44, 10.2021, p. 16053-16066.

Publications: Contribution to journalArticlePeer Reviewed


Effects of N-terminus modified Hx-amides on DNA binding affinity, sequence specificity, cellular uptake, and gene expression. / Kiakos, Konstantinos (Corresponding author); Satam, Vijay; Patil, Pravin C. et al.
In: Bioorganic & Medicinal Chemistry Letters, Vol. 47, 128158, 01.09.2021.

Publications: Contribution to journalArticlePeer Reviewed


Modified amino-dextrans as carriers of Gd-chelates for retrograde transport and visualization of peripheral nerves by magnetic resonance imaging (MRI). / Pashkunova-Martic, Irena (Corresponding author); Manzano-Szalai, Krisztina; Friske, Joachim et al.
In: Journal of Inorganic Biochemistry, Vol. 222, 111495, 09.2021.

Publications: Contribution to journalArticlePeer Reviewed


Structure-Activity Relationships of Triple-Action Platinum(IV) Prodrugs with Albumin-Binding Properties and Immunomodulating Ligands. / Fronik, Philipp; Poetsch, Isabella; Kastner, Alexander et al.
In: Journal of Medicinal Chemistry, Vol. 64, No. 16, 26.08.2021, p. 12132-12151.

Publications: Contribution to journalArticlePeer Reviewed


Hunting for bis-bibenzyls in Primula veris subsp. macrocalyx (Bunge) Lüdi: Organ-specific accumulation and cytotoxic activity. / Bukvicki, Danka (Corresponding author); Kovtonyuk, Nataliya K.; Legin, Anton A. et al.
In: Phytochemistry Letters, Vol. 44, 08.2021, p. 90-97.

Publications: Contribution to journalArticlePeer Reviewed


Thermodynamic Genome-Scale Metabolic Modeling of Metallodrug Resistance in Colorectal Cancer. / Herrmann, Helena A.; Rusz, Mate; Baier, Dina et al.
In: Cancers, Vol. 13, No. 16, 4130, 08.2021.

Publications: Contribution to journalArticlePeer Reviewed


Morpho-metabotyping the oxidative stress response. / Rusz, Mate; Del Favero, Giorgia; El Abiead, Yasin et al.
In: Scientific Reports, Vol. 11, No. 1, 15471, 29.07.2021.

Publications: Contribution to journalArticlePeer Reviewed


Toward a deeper and simpler understanding of serum protein-mediated transformations of magnetic nanoparticles by ICP-MS. / Kuznetsova, Olga; Jarosz, Maciej; Keppler, Bernhard K. et al.
In: Talanta, Vol. 229, 122287, 01.07.2021.

Publications: Contribution to journalArticlePeer Reviewed


Complex formation of an estrone-salicylaldehyde semicarbazone hybrid with copper(II) and gallium(III): Solution equilibria and biological activity. / Enyedy, Eva A. (Corresponding author); Petrasheuskaya, Tatsiana; Kiss, Marton A. et al.
In: Journal of Inorganic Biochemistry, Vol. 220, 111468, 07.2021.

Publications: Contribution to journalArticlePeer Reviewed


Establishing electron diffraction in chemical crystallography. / Gruene, Tim (Corresponding author); Holstein, Julian J. (Corresponding author); Clever, Guido H. et al.
In: Nature reviews chemistry, Vol. 5, No. 9, 07.2021, p. 660–668.

Publications: Contribution to journalReviewPeer Reviewed


Multifunctional Pt(iv) prodrug candidates featuring the carboplatin core and deferoxamine. / Harringer, Sophia; Hejl, Michaela; Enyedy, Eva A. et al.
In: Dalton Transactions, Vol. 50, No. 23, 18.05.2021, p. 8167-8178.

Publications: Contribution to journalArticlePeer Reviewed


Micro-droplet-based calibration for quantitative elemental bioimaging by LA-ICPMS. / Schweikert, Andreas; Theiner, Sarah (Corresponding author); Wernitznig, Debora et al.
In: Analytical and Bioanalytical Chemistry, Vol. 414, No. 1, 05.05.2021, p. 485–495.

Publications: Contribution to journalArticlePeer Reviewed


Current trends and challenges in analysis and characterization of engineered nanoparticles in seawater. / Timerbaev, Andrei R. (Corresponding author); Kuznetsova, Olga; Keppler, Bernhard K.
In: Talanta, Vol. 226, 122201, 05.2021.

Publications: Contribution to journalReviewPeer Reviewed


Mass spectrometry techniques for imaging and detection of metallodrugs. / Theiner, Sarah; Schoeberl, Anna; Schweikert, Andreas et al.
In: Current opinion in chemical biology, Vol. 61, 04.2021, p. 123-134.

Publications: Contribution to journalReviewPeer Reviewed


Development of a cobalt(iii)-based ponatinib prodrug system. / Mathuber, Marlene; Gutmann, Michael; La Franca, Mery et al.
In: Inorganic Chemistry Frontiers, Vol. 8, No. 10, 30.03.2021, p. 2468-2485.

Publications: Contribution to journalArticlePeer Reviewed


Interaction with Ribosomal Proteins Accompanies Stress Induction of the Anticancer Metallodrug BOLD-100/KP1339 in the Endoplasmic Reticulum. / Neuditschko, Benjamin; Legin, Anton A.; Baier, Dina et al.
In: Angewandte Chemie (International Edition), Vol. 60, No. 10, 01.03.2021, p. 5063-5068.

Publications: Contribution to journalArticlePeer Reviewed


Doubly derivatized poly(lactide)-albumin nanoparticles as blood vessel-targeted transport device for magnetic resonance imaging (MRI). / Pashkunova-Martic, Irena (Corresponding author); Kremser, Christian; Talasz, Heribert et al.
In: Journal of Nanoparticle Research, Vol. 23, No. 2, 51, 18.02.2021.

Publications: Contribution to journalArticlePeer Reviewed