o. Univ.-Prof. Dr. Dr. Bernhard Keppler

Email: bernhard.keppler@univie.ac.at
Phone: +43-1-4277-52602

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Publications



The gallium complex KP46 sensitizes resistant leukemia cells and overcomes Bcl-2-induced multidrug resistance in lymphoma cells via upregulation of Harakiri and downregulation of XIAP in vitro. / Wilke, Nicola L.; Abodo, Liliane Onambele; Frias, Corazon et al.
In: Biomedicine and Pharmacotherapy, Vol. 156, 113974, 12.2022.

Publications: Contribution to journalArticlePeer Reviewed


Novel Salinomycin-Based Paramagnetic Complexes-First Evaluation of Their Potential Theranostic Properties. / Pashkunova-Martic, Irena (Corresponding author); Kukeva, Rositsa; Stoyanova, Radostina et al.
In: Pharmaceutics, Vol. 14, No. 11, 2319, 11.2022.

Publications: Contribution to journalArticlePeer Reviewed


Oxoplatin-Based Pt(IV) Lipoate Complexes and Their Biological Activity. / Liu, Xiao; Barth, Marie-Christin; Cseh, Klaudia et al.
In: Chemistry & Biodiversity, Vol. 19, No. 10, e202200695, 10.2022.

Publications: Contribution to journalArticlePeer Reviewed


Thiosemicarbazone Derivatives Developed to Overcome COTI-2 Resistance. / Posa, Vivien; Stefanelli, Alessia; Nunes, Julia H. Bormio et al.
In: Cancers, Vol. 14, No. 18, 4455, 09.2022.

Publications: Contribution to journalArticlePeer Reviewed


Quantification in bioimaging by LA-ICPMS - Evaluation of isotope dilution and standard addition enabled by micro-droplets. / Schweikert, Andreas; Theiner, Sarah (Corresponding author); Sala, Martin et al.
In: Analytica Chimica Acta, Vol. 1223, 340200, 29.08.2022.

Publications: Contribution to journalArticlePeer Reviewed


Current Developments of N-Heterocyclic Carbene Au(I)/Au(III) Complexes toward Cancer Treatment. / Tialiou, Alexia; Chin, Jia Min (Corresponding author); Keppler, Bernhard K. et al.
In: Biomedicines, Vol. 10, No. 6, 1417, 06.2022.

Publications: Contribution to journalReviewPeer Reviewed


The coordination modes of (thio)semicarbazone copper(II) complexes strongly modulate the solution chemical properties and mechanism of anticancer activity. / Posa, Vivien; Hajdu, Balint; Toth, Gabor et al.
In: Journal of Inorganic Biochemistry, Vol. 231, 111786, 06.2022.

Publications: Contribution to journalArticlePeer Reviewed


Comparative Effects of Deferiprone and Salinomycin on Lead-Induced Disturbance in the Homeostasis of Intrarenal Essential Elements in Mice. / Gluhcheva, Yordanka; Pashkunova-Martic, Irena; Schaier, Martin et al.
In: International Journal of Molecular Sciences, Vol. 23, No. 8, 4368, 15.04.2022.

Publications: Contribution to journalArticlePeer Reviewed


A platinum(IV) prodrug strategy to overcome glutathione-based oxaliplatin resistance. / Fronik, Philipp; Gutmann, Michael; Vician, Petra et al.
In: Communications Chemistry, Vol. 5, No. 1, 46, 06.04.2022.

Publications: Contribution to journalArticlePeer Reviewed


Solution speciation and human serum protein binding of indium(III) complexes of 8-hydroxyquinoline, deferiprone and maltol. / Domotor, Orsolya (Corresponding author); Keppler, Bernhard K.; Enyedy, Eva A.
In: Journal of Biological Inorganic Chemistry, Vol. 27, No. 3, 04.2022, p. 315-328.

Publications: Contribution to journalArticlePeer Reviewed


Versatile analytical methodology for evaluation of drug-like properties of potentially multi-targeting anticancer metallodrugs. / Foteeva, Lidia S.; Nosova, Yulia N.; Nazarov, Alexey A. et al.
In: Analytical Sciences, Vol. 38, No. 3, 03.2022, p. 627-632.

Publications: Contribution to journalArticlePeer Reviewed


Systematic Study on the Cytotoxic Potency of Commonly Used Dimeric Metal Precursors in Human Cancer Cell Lines. / Geisler, Heiko; Harringer, Sophia; Wenisch, Dominik et al.
In: ChemistryOpen, Vol. 11, No. 7, e202200019, 24.02.2022.

Publications: Contribution to journalArticlePeer Reviewed


The Anticancer Ruthenium Compound BOLD-100 Targets Glycolysis and Generates a Metabolic Vulnerability towards Glucose Deprivation. / Baier, Dina; Schönhacker-Alte, Beatrix; Rusz, Mate et al.
In: Pharmaceutics, Vol. 14, No. 2, 238, 20.01.2022.

Publications: Contribution to journalArticlePeer Reviewed


Organometallic Receptors and Conjugates With Biomolecules in Bioorganometallic Chemistry. / Neuditschko, Benjamin; Keppler, Bernhard K.; Gerner, Christopher et al.
Comprehensive Organometallic Chemistry IV: Volume 1-15. Vol. 1-15 Elsevier, 2022. p. 183-205.

Publications: Contribution to bookChapterPeer Reviewed


Novel oxaliplatin(IV) complexes conjugated with ligands bearing pendant 1,2-dithiolane/1,2-diselenolane/cyclopentyl motifs. / Liu, Xiao; Wenisch, Dominik; Barth, Marie-Christin et al.
In: Dalton Transactions, Vol. 51, No. 44, 2022, p. 16824-16835.

Publications: Contribution to journalArticlePeer Reviewed


Elemental analysis: an important purity control but prone to manipulations. / Kandioller, Wolfgang; Theiner, Johannes; Keppler, Bernhard K. et al.
In: Inorganic Chemistry Frontiers, Vol. 9, No. 3, 12.2021, p. 412-416.

Publications: Contribution to journalArticlePeer Reviewed


Water-soluble trithiolato-bridged dinuclear ruthenium(II) and osmium(II) arene complexes with bisphosphonate functionalized ligands as anticancer organometallics. / Riedl, Christoph A.; Rosner, Alexander; Harringer, Sophia et al.
In: Journal of Inorganic Biochemistry, Vol. 225, 111618, 12.2021.

Publications: Contribution to journalArticlePeer Reviewed


Albumin-targeting of an oxaliplatin-releasing platinum(iv) prodrug results in pronounced anticancer activity due to endocytotic drug uptake in vivo. / Schueffl, Hemma; Theiner, Sarah; Hermann, Gerrit et al.
In: Chemical Science, Vol. 12, No. 38, 14.10.2021, p. 12587-12599.

Publications: Contribution to journalArticlePeer Reviewed