o. Univ.-Prof. Dr. Dr. Bernhard Keppler

Email: bernhard.keppler@univie.ac.at
Phone: +43-1-4277-52602

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Publications


Showing entries 121 - 140 out of 688
Fine-Tuning the Activation Mode of an 1,3-Indandione-Based Ruthenium(II)-Cymene Half-Sandwich Complex by Variation of Its Leaving Group. / Mokesch, Stephan; Schwarz, Daniela; Hejl, Michaela et al.
In: Molecules, Vol. 24, No. 13, 2373, 01.07.2019.

Publications: Contribution to journalArticlePeer Reviewed


Subcellular Duplex DNA and G-Quadruplex Interaction Profiling of a Hexagonal Pt-II Metallacycle. / Domarco, Olaya; Kieler, Claudia; Pirker, Christine et al.
In: Angewandte Chemie (International Edition), Vol. 58, No. 24, 11.06.2019, p. 8007-8012.

Publications: Contribution to journalArticlePeer Reviewed


First-in-class ruthenium anticancer drug (KP1339/IT-139) induces an immunogenic cell death signature in colorectal spheroids in vitro. / Wernitznig, Debora (Corresponding author); Kiakos, Konstantinos; Del Favero, Giorgia et al.
In: Metallomics: integrated biometal science, Vol. 11, No. 6, 01.06.2019, p. 1044-1048.

Publications: Contribution to journalArticlePeer Reviewed


Synthesis, characterization, lipophilicity and cytotoxic properties of novel bis(carboxylato)oxalatobis(1-propylamine)platinum(IV) complexes. / Hizal, Selin; Hejl, Michaela; Jakupec, Michael A. et al.
In: Inorganica Chimica Acta, Vol. 491, 01.06.2019, p. 76-83.

Publications: Contribution to journalArticlePeer Reviewed


A Dogma in Doubt: Hydrolysis of Equatorial Ligands of Pt-IV Complexes under Physiological Conditions. / Kastner, Alexander; Poetsch, Isabella; Mayr, Josef et al.
In: Angewandte Chemie (International Edition), Vol. 58, No. 22, 27.05.2019, p. 7464-7469.

Publications: Contribution to journalArticlePeer Reviewed


Synthesis, characterization, cytotoxic activity, and F-19 NMR spectroscopic investigations of (OC-6-33)-diacetato(ethane-1,2-diamine)bis(3,3,3-trifluoropropanoato)platinum(IV) and its platinum(II) counterpart. / Hoefer, Doris; Cseh, Klaudia; Hejl, Michaela et al.
In: Inorganica Chimica Acta, Vol. 490, 01.05.2019, p. 190-199.

Publications: Contribution to journalArticlePeer Reviewed


Challenges and Chances in the Preclinical to Clinical Translation of Anticancer Metallodrugs. / Pötsch, Isabella; Baier, Dina; Keppler, Bernhard et al.
Metal-based Anticancer Agents . ed. / Angela Casini; Anne Vessieres; Samuel M. Meier-Menches. Royal Society of Chemistry, 2019. p. 308 - 347 (RSC Metallobiology; No. 14, Vol. 2019-January).

Publications: Contribution to bookChapterPeer Reviewed


A simple assay for probing transformations of superparamagnetic iron oxide nanoparticles in human serum. / Kuznetsova, Olga; Reshetnikova, Irina S.; Shtykov, Sergei N. et al.
In: Chemical Communications, Vol. 55, No. 29, 14.04.2019, p. 4270-4272.

Publications: Contribution to journalArticlePeer Reviewed


Analytical methodology for studying cellular uptake, processing and localization of gold nanoparticles. / Matczuk, Magdalena; Ruzik, Lena; Aleksenko, Svetlana S. et al.
In: Analytica Chimica Acta, Vol. 1052, 04.04.2019, p. 1-9.

Publications: Contribution to journalReviewPeer Reviewed


Mercury, silver, selenium and other trace elements in three cyprinid fish species from the Vaal Dam, South Africa, including implications for fish consumers. / Plessl, Christof; Gilbert, Beric M.; Sigmund, Martin F. et al.
In: Science of the Total Environment, Vol. 659, 01.04.2019, p. 1158-1167.

Publications: Contribution to journalArticlePeer Reviewed


Natural iron fertilization of the coastal ocean by "blackwater rivers". / Krachler, Regina (Corresponding author); Krachler, Rudolf; Valda, Alexander et al.
In: Science of the Total Environment, Vol. 656, 15.03.2019, p. 952-958.

Publications: Contribution to journalArticlePeer Reviewed


Bacterial ghosts as adjuvant to oxaliplatin chemotherapy in colorectal carcinomatosis. / Groza, D.; Gehrig, S.; Dinhof, C. et al.
In: European Journal of Cancer, Vol. 110, No. S1, 03.2019, p. S23-S24.

Publications: Contribution to journalMeeting abstract/Conference paperPeer Reviewed


Synthesis, Characterization, Cytotoxicity, and Time-Dependent NMR Spectroscopic Studies of (SP-4-3)-Oxalato[(1R,2R,4R/1S,2S,4S)-(4-trifluoromethyl-cyclohexane-1,2-diamine)]platinum(II). / Hizal, Selin; Hejl, Michaela; Jungmann, Christoph et al.
In: European Journal of Inorganic Chemistry, Vol. 2019, No. 6, 14.02.2019, p. 856-864.

Publications: Contribution to journalArticlePeer Reviewed


Metal Drugs and the Anticancer Immune Response. / Englinger, Bernhard; Pirker, Christine; Heffeter, Petra et al.
In: Chemical Reviews, Vol. 119, No. 2, 23.01.2019, p. 1519-1624.

Publications: Contribution to journalReviewPeer Reviewed


Synthesis and biological evaluation of biotin-conjugated anticancer thiosemicarbazones and their iron(III) and copper(II) complexes. / Kallus, Sebastian; Uhlik, Lukas; van Schoonhoven, Sushilla et al.
In: Journal of Inorganic Biochemistry, Vol. 190, 01.2019, p. 85-97.

Publications: Contribution to journalArticlePeer Reviewed


Synthesis, Characterization and in vitro Studies of a Cathepsin B-Cleavable Prodrug of the VEGFR Inhibitor Sunitinib. / Karnthaler-Benbakka, Claudia; Koblmueller, Bettina; Mathuber, Marlene et al.
In: Chemistry & Biodiversity, Vol. 16, No. 1, e1800520, 01.2019.

Publications: Contribution to journalArticlePeer Reviewed


Anticancer Thiosemicarbazones: Chemical Properties, Interaction with Iron Metabolism, and Resistance Development. / Heffeter, Petra (Corresponding author); Pape, Veronika F. S.; Enyedy, Eva A. et al.
In: Antioxidants and Redox Signaling, Vol. 30, No. 8, 2019, p. 1062-1082.

Publications: Contribution to journalArticlePeer Reviewed


New Variations on the Theme of Gold(III) C N N Cyclometalated Complexes as Anticancer Agents: Synthesis and Biological Characterization. / Carboni, Silvia; Zucca, Antonio; Stoccoro, Sergio et al.
In: Inorganic Chemistry, Vol. 57, No. 23, 03.12.2018, p. 14852-14865.

Publications: Contribution to journalArticlePeer Reviewed


Development and Validation of Liquid Chromatography-Based Methods to Assess the Lipophilicity of Cytotoxic Platinum(IV) Complexes. / Klose, Matthias H. M.; Theiner, Sarah; Varbanov, Hristo P. et al.
Unconventional Anticancer Metallodrugs and Strategies to Improve their Pharmacological Profile. ed. / Maria Contel. Vol. 6 4. ed. Basel: Multi-disciplinary digital publishing institute (MDPI), 2018. p. 71-84 130 (Inorganics).

Publications: Contribution to bookChapterPeer Reviewed


Biological activity of Pt-IV prodrugs triggered by riboflavin-mediated bioorthogonal photocatalysis. / Alonso-de Castro, Silvia; Terenzi, Alessio; Hager, Sonja et al.
In: Scientific Reports, Vol. 8, No. 1, 17198, 21.11.2018.

Publications: Contribution to journalArticlePeer Reviewed


Showing entries 121 - 140 out of 688