2020

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1,4-Disubstituted 1,2,3-Triazoles as Amide Bond Surrogates for the Stabilisation of Linear Peptides with Biological Activity
Recnik, L-M., Kandioller, W. & Mindt, T. L.
Molecules (2020) 25, 16, 3576

Single Peptide Backbone Surrogate Mutations to Regulate Angiotensin GPCR Subtype Selectivity
Vrettos, E., Valverde, I. E., Mascarin, A., Pallier, P. N., Cerofolini, L., Fragai, M., Parigi, G., Hirmiz, B., Bekas, N., Grob, N. M., Shaye, H., Del Borgo, M., Aguilar, M., Magnani, F., Syed, N., Crook, T., Waqif, E., Ghazaly, E., Cherezov, V., Widdop, R. E., Luchinat, C., Michael-Titus, A. T., Mindt, T. L., Tzakos, A. G. & Stylos, E. K.
Chemistry: A European Journal (2020) 26, 47, 10690-10694

Radiolabelling of the octadentate chelators DFO* and oxoDFO* with zirconium-89 and gallium-68
Brandt, M., Cowell, J., Aulsebrook, M. L., Gasser, G. & Mindt, T. L.
Journal of Biological Inorganic Chemistry (2020) 25, 789–796

Sorbitol as a Polar Pharmacological Modifier to Enhance the Hydrophilicity of 99mTc-Tricarbonyl-Based Radiopharmaceuticals
Giammei, C., Balber, T., Benčurová, K., Cardinale, J., Berroterán-Infante, N., Brandt, M., Jouini, N., Hacker, M., Mitterhauser, M. & Mindt, T. L.
Molecules (2020) 25, 11, 2680

Design of Radiolabeled Analogs of Minigastrin by Multiple Amide-to-Triazole Substitutions
Grob, N. M., Schmid, S., Schibli, R., Behe, M. & Mindt, T. L.
Journal of Medicinal Chemistry (2020) 63, 9, 4496-4505

Triazolo-Peptidomimetics: Novel Radiolabeled Minigastrin Analogs for Improved Tumor Targeting
Grob, N. M., Haussinger, D., Deupi, X., Schibli, R., Behe, M. & Mindt, T. L.
Medicinal Chemistry (2020) 63, 9, 4484-4495